产品名称

英文名称：Sarpogrelate Hydrochloride

同义词

sarpogrelate hydrochloride、135159-51-2、Sarpogrelate HCl、Anplag、MCI-9042、Mci 9042、Sarpogrelate (hydrochloride)、Sarpogrelate hydrochloride [JAN]、Sarpogrelatehydrochloride、FQN8N8QP1B、DTXSID8046662、CHEMBL541829、4-[1-(dimethylamino)-3-[2-[2-(3-methoxyphenyl)et、盐酸沙格雷酯

产品性质

CAS编号：135159-51-2

分子式：C24H31NO6.HCl

分子量：465.97

MDL号：MFCD00887582

PubChem编号：444005

别名：盐酸沙格雷酯

英文别名：sarpogrelate hydrochloride|135159-51-2|Sarpogrelate HCl|Anplag|MCI-9042|Mci 9042|Sarpogrelate (hydrochloride)|Sarpogrelate hydrochloride [JAN]|Sarpogrelatehydrochloride|FQN8N8QP1B|DTXSID8046662|CHEMBL541829|4-[1-(dimethylamino)-3-[2-[2-(3-methoxyphenyl)et

规格或纯度：≥98%

英文名称：Sarpogrelate Hydrochloride

生化机理：选择性5-HT2A受体拮抗剂（5-HT2A，5-HT2C和5-HT2B受体的pKi值分别为8.52、7.43和6.57）。对5-HT1、5-HT3、5-HT4H1，H2，M3，α1-肾上腺素能，α2-肾上腺素能和β-肾上腺素能受体显示选择性。在体内显示出心脏保护活性。

运输条件：常规运输

备注：卖完停产，不再备货

产品介绍：Sarpogrelate hydrochloride (盐酸沙格雷酯; MCI-9042) 是5-HT2拮抗剂，可用作抗血小板类化合物。Soluble in water (25 mM), DMSO (100 mM), and methanol.Sarpogrelate(MCI-9042) hydrochloride, a selective 5-HT2 antagonist, has been widely used as an anti-platelet agent for the treatment of PAD.Soluble in water (25 mM), DMSO (100 mM), and methanol.

PubChem SID：488189819

IUPAC Name：4-[1-(dimethylamino)-3-[2-[2-(3-methoxyphenyl)ethyl]phenoxy]propan-2-yl]oxy-4-oxobutanoic acid;hydrochloride

INCHI：InChI=1S/C24H31NO6.ClH/c1-25(2)16-21(31-24(28)14-13-23(26)27)17-30-22-10-5-4-8-19(22)12-11-18-7-6-9-20(15-18)29-3;/h4-10,15,21H,11-14,16-17H2,1-3H3,(H,26,27);1H

InChi Key：POQBIDFFYCYHOB-UHFFFAOYSA-N

Canonical SMILES：CN(C)CC(COC1=CC=CC=C1CCC2=CC(=CC=C2)OC)OC(=O)CCC(=O)O.Cl

Isomeric SMILES：CN(C)CC(COC1=CC=CC=C1CCC2=CC(=CC=C2)OC)OC(=O)CCC(=O)O.Cl

WGK Germany：3

PubChem CID：444005

溶解性：溶于water, 最高浓度 (mg/mL) 11.65, 最高浓度(mM) 25；溶于DMSO, 最高浓度 (mg/mL) 46.6, 最高浓度(mM) 100

象形图：

信号词：Warning

危险声明：H302 Harmful if swallowedH400 Very toxic to aquatic life

预防措施声明：P273,P501,P264,P270,P391,P330,P301+P317

产品包装