产品名称

英文名称：Tianeptine Sodium Salt Hydrate

同义词

Tianeptine sodium、30123-17-2、Tianeptine sodium salt、Stablon、Coaxil、Tatinol、Tianeptine (sodium salt)、Tianeptine sodium salt hydrate、169293-32-7、(+)-Tianeptine Monosodium Salt、Tianeptine sodium, (+)-、sodium;7-[(3-chloro-6-methyl-5,5-dioxo-11H-benzo[c][2,1]b、噻奈普汀钠水合物、7-[[3-氯-6,11-二氢-6-甲基二苯并[c,f][1,2]硫氮杂卓-11-基]氨基]庚酸S,S-二氧化物钠盐水合物

产品性质

CAS编号：30123-17-2

分子式：C21H24ClN2NaO4S·xH2O

分子量：458.93(anhydrous basis)

MDL号：MFCD00879851

PubChem编号：23663953

别名：噻奈普汀钠水合物|7-[[3-氯-6,11-二氢-6-甲基二苯并[c,f][1,2]硫氮杂卓-11-基]氨基]庚酸S,S-二氧化物钠盐水合物

英文别名：Tianeptine sodium|30123-17-2|Tianeptine sodium salt|Stablon|Coaxil|Tatinol|Tianeptine (sodium salt)|Tianeptine sodium salt hydrate|169293-32-7|(+)-Tianeptine Monosodium Salt|Tianeptine sodium, (+)-|sodium;7-[(3-chloro-6-methyl-5,5-dioxo-11H-benzo[c][2,1]b

规格或纯度：>98.0%(HPLC)

英文名称：Tianeptine Sodium Salt Hydrate

生化机理：选择性5-HT吸收促进剂。在体内显示出抗抑郁，镇痛，神经保护和认知增强作用。口服具有活性

储存温度：-20°C储存

运输条件：超低温冰袋运输

备注：如果有可能，您尽量在使用的当天配置溶液，并在当天使用完它。但是，如果您需要预先配制储备溶液，我们建议您将溶液等份保存在-20°C的密封小瓶中。通常，它们最多可以使用一个月。在使用前和打开样品瓶之前，我们建议您让您的产品在室温下平衡至少1小时。需要更多关于溶解度，用法和处理的建议吗？请访问我们的常见问题（FAQ）页面以获取更多详细信息。

产品介绍：Sodium has been assayed as a steatosis-positive inducer in HepG2 cells. Tianeptine has also been used to study effects on rats exposed to swim endurance tests (SETs). This study reported that tianeptine increased swimming time in rats undergoing SET. Moreover, tianeptine also increased total cholesterol and LDL, while triglyceride levels were decreased. Thus, tianeptine may be involved in the pathogenesis of metabolic syndrome.

IUPAC Name：sodium;7-[(3-chloro-6-methyl-5,5-dioxo-11H-benzo[c][2,1]benzothiazepin-11-yl)amino]heptanoate

INCHI：InChI=1S/C21H25ClN2O4S.Na/c1-24-18-9-6-5-8-16(18)21(23-13-7-3-2-4-10-20(25)26)17-12-11-15(22)14-19(17)29(24,27)28;/h5-6,8-9,11-12,14,21,23H,2-4,7,10,13H2,1H3,(H,25,26);/q;+1/p-1

InChi Key：ZLBSUOGMZDXYKE-UHFFFAOYSA-M

Canonical SMILES：CN1C2=CC=CC=C2C(C3=C(S1(=O)=O)C=C(C=C3)Cl)NCCCCCCC(=O)[O-].[Na+]

Isomeric SMILES：CN1C2=CC=CC=C2C(C3=C(S1(=O)=O)C=C(C=C3)Cl)NCCCCCCC(=O)[O-].[Na+]

关联CAS：72797-41-2

PubChem CID：23663953

溶解性：可溶于甲醇

熔点：184 °C

象形图：

信号词：Danger

危险声明：H301 Toxic if swallowedH373 Causes damage to organs through prolonged or repeated exposureH302 Harmful if swallowedH312 Harmful in contact with skinH332 Harmful if inhaledH361 Suspected of damaging fertility or the unborn childH362 May cause harm to breast-fed children

预防措施声明：P261,P280,P302+P352,P321,P405,P501,P264,P260,P271,P270,P304+P340,P362+P364,P330,P263,P203,P301+P316,P301+P317,P318,P317,P319

Merck Index：9420

产品包装